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ALDH3A1

receptor: AhRTier 1

Drug substrates

cyclophosphamide; doxorubicin; fluorouracil

refs: 24677340

CAMIP causal chains

AhR

Reduced AhR-mediated induction of ALDH3A1 would lower ALDH3A1-mediated oxidation of aldophosphamide; increased retention of the active intermediate may sensitise tumour cells to cyclophosphamide.

Drug context: cyclophosphamide; doxorubicin; fluorouracil

Scored variants near ALDH3A1

chr17:19,637,984..19,848,298, gene body plus 100 kb. Showing the strongest 200 by effect size.

Variant Position PXR FXR AhR AF
chr17_19648971_C_Gchr17:196489711.0000.0480.259—   
chr17_19648978_C_Gchr17:196489781.0001.0000.565—   
chr17_19648930_C_Achr17:196489301.0000.3220.341—   
chr17_19649058_C_Gchr17:196490580.9980.1420.3120.0046%
chr17_19648985_T_Cchr17:19648985-0.972-0.787-0.600—   
chr17_19648985_T_Achr17:19648985-0.955-0.792-0.671—   
chr17_19648985_T_Gchr17:19648985-0.935-0.769-0.506—   
chr17_19648862_C_Gchr17:19648862-0.885-0.482-0.176—   
chr17_19648984_G_Achr17:19648984-0.882-0.670-0.494—   
chr17_19648981_G_Achr17:196489810.8750.9110.318—   
chr17_19648977_G_Achr17:19648977-0.872-0.553-0.576—   
chr17_19648984_G_Tchr17:19648984-0.869-0.614-0.435—   
chr17_19648981_G_Cchr17:19648981-0.865-0.637-0.518—   
chr17_19648804_G_Achr17:196488040.8320.4800.282—   
chr17_19648860_G_Cchr17:196488600.8320.1980.365—   
chr17_19648977_G_Tchr17:19648977-0.812-0.647-0.471—   
chr17_19648980_C_Gchr17:19648980-0.802-0.528-0.400—   
chr17_19648799_A_Gchr17:19648799-0.792-0.480-0.094—   
chr17_19649017_C_Achr17:196490170.7920.7660.535—   
chr17_19648982_A_Gchr17:19648982-0.775-0.576-0.318—   
chr17_19648931_C_Achr17:196489310.7690.1850.435—   
chr17_19648792_G_Cchr17:19648792-0.765-0.325-0.153—   
chr17_19648982_A_Cchr17:19648982-0.752-0.566-0.271—   
chr17_19648980_C_Achr17:19648980-0.742-0.500-0.471—   
chr17_19648865_C_Gchr17:196488650.7320.0150.082—   
chr17_19648984_G_Cchr17:19648984-0.722-0.500-0.365—   
chr17_19648996_C_Achr17:196489960.7220.6830.329—   
chr17_19648820_G_Cchr17:19648820-0.709-0.173-0.059—   
chr17_19649017_C_Gchr17:196490170.7050.7440.359—   
chr17_19648982_A_Tchr17:19648982-0.689-0.513-0.306—   
chr17_19648799_A_Tchr17:19648799-0.686-0.662-0.141—   
chr17_19648923_C_Achr17:196489230.6790.4060.294—   
chr17_19648782_G_Tchr17:196487820.1400.2161.000—   
chr17_19648983_A_Tchr17:19648983-0.662-0.538-0.282—   
chr17_19648865_C_Achr17:196488650.6520.0910.082—   
chr17_19648980_C_Tchr17:19648980-0.649-0.416-0.365—   
chr17_19648977_G_Cchr17:19648977-0.636-0.548-0.259—   
chr17_19648983_A_Cchr17:19648983-0.626-0.363-0.294—   
chr17_19649025_A_Tchr17:19649025-0.626-0.579-0.129—   
chr17_19648946_C_Gchr17:196489460.6220.2010.318—   
chr17_19648981_G_Tchr17:19648981-0.619-0.487-0.471—   
chr17_19649023_C_Tchr17:196490230.6090.6240.265—   
chr17_19649028_T_Achr17:19649028-0.609-0.520-0.259—   
chr17_19648877_G_Achr17:19648877-0.606-0.363-0.3530.0013%
chr17_19648877_G_Tchr17:19648877-0.606-0.571-0.529—   
chr17_19648987_C_Gchr17:19648987-0.602-0.475-0.388—   
chr17_19648930_C_Tchr17:196489300.5890.1500.165—   
chr17_19648987_C_Achr17:19648987-0.579-0.363-0.435—   
chr17_19648923_C_Gchr17:196489230.5660.2210.306—   
chr17_19648928_T_Cchr17:19648928-0.386-0.404-1.000—   
chr17_19648990_C_Gchr17:19648990-0.566-0.343-0.471—   
chr17_19649056_G_Achr17:19649056-0.566-0.272-0.412—   
chr17_19648859_A_Gchr17:196488590.5590.2990.047—   
chr17_19648836_T_Cchr17:196488360.5520.4310.1880.0046%
chr17_19649076_G_Achr17:196490760.5520.5860.876—   
chr17_19648979_T_Cchr17:19648979-0.549-0.371-0.294—   
chr17_19648877_G_Cchr17:19648877-0.536-0.305-0.200—   
chr17_19649025_A_Gchr17:19649025-0.532-0.525-0.082—   
chr17_19648932_C_Tchr17:196489320.5290.0960.224—   
chr17_19648843_T_Gchr17:19648843-0.526-0.249-0.012—   
chr17_19648939_C_Achr17:196489390.5260.3600.247—   
chr17_19648930_C_Gchr17:196489300.5160.1800.259—   
chr17_19649023_C_Gchr17:19649023-0.512-0.381-0.259—   
chr17_19648983_A_Gchr17:19648983-0.509-0.472-0.200—   
chr17_19648861_A_Cchr17:196488610.5060.2540.188—   
chr17_19649024_G_Cchr17:19649024-0.506-0.442-0.159—   
chr17_19648792_G_Tchr17:19648792-0.499-0.185-0.165—   
chr17_19648865_C_Tchr17:196488650.4990.056-0.071<0.001%
chr17_19648878_G_Achr17:19648878-0.499-0.322-0.318—   
chr17_19648925_C_Tchr17:196489250.4990.2180.153—   
chr17_19648979_T_Gchr17:19648979-0.496-0.299-0.212<0.001%
chr17_19649024_G_Tchr17:19649024-0.496-0.467-0.312—   
chr17_19648988_G_Achr17:196489880.4930.3200.188—   
chr17_19648987_C_Tchr17:19648987-0.489-0.373-0.412<0.001%
chr17_19648991_G_Cchr17:19648991-0.483-0.279-0.318—   
chr17_19649023_C_Achr17:19649023-0.479-0.335-0.312—   
chr17_19648942_G_Tchr17:196489420.4760.2160.176—   
chr17_19648921_C_Achr17:19648921-0.473-0.500-0.282—   
chr17_19648785_C_Tchr17:19648785-0.469-0.437-0.235—   
chr17_19648881_G_Achr17:19648881-0.469-0.305-0.212—   
chr17_19648922_T_Cchr17:19648922-0.243-0.165-0.824—   
chr17_19648988_G_Tchr17:19648988-0.463-0.391-0.353—   
chr17_19648839_T_Gchr17:19648839-0.459-0.1780.035—   
chr17_19648863_A_Cchr17:19648863-0.459-0.1980.000—   
chr17_19648878_G_Cchr17:19648878-0.459-0.264-0.329—   
chr17_19648784_A_Tchr17:19648784-0.456-0.124-0.212—   
chr17_19648876_A_Tchr17:19648876-0.456-0.274-0.200—   
chr17_19649027_C_Tchr17:19649027-0.456-0.391-0.259—   
chr17_19648880_G_Tchr17:19648880-0.449-0.259-0.212—   
chr17_19648920_C_Achr17:19648920-0.443-0.282-0.129—   
chr17_19648777_C_Achr17:19648777-0.439-0.1500.000—   
chr17_19648904_A_Cchr17:19648904-0.439-0.320-0.165—   
chr17_19648908_G_Cchr17:19648908-0.439-0.447-0.176—   
chr17_19648988_G_Cchr17:19648988-0.436-0.431-0.2710.0013%
chr17_19649085_G_Tchr17:196490850.436-0.1700.153—   
chr17_19648829_G_Cchr17:196488290.4330.3350.165—   
chr17_19648853_C_Gchr17:196488530.4330.2690.212—   
chr17_19648880_G_Cchr17:19648880-0.433-0.272-0.165—   
chr17_19648986_C_Gchr17:19648986-0.433-0.287-0.176—   
chr17_19648878_G_Tchr17:19648878-0.426-0.213-0.318—   
chr17_19648919_G_Tchr17:196489190.4190.1780.000—   
chr17_19648925_C_Gchr17:196489250.4160.0910.141—   
chr17_19648880_G_Achr17:19648880-0.413-0.256-0.259—   
chr17_19648892_G_Tchr17:19648892-0.409-0.327-0.447—   
chr17_19649024_G_Achr17:19649024-0.409-0.363-0.306—   
chr17_19649028_T_Gchr17:19649028-0.409-0.426-0.112—   
chr17_19648862_C_Tchr17:19648862-0.406-0.228-0.094—   
chr17_19648931_C_Gchr17:196489310.4060.0890.235—   
chr17_19648793_G_Achr17:19648793-0.403-0.1320.000<0.001%
chr17_19648794_C_Achr17:19648794-0.403-0.058-0.259—   
chr17_19648881_G_Tchr17:19648881-0.403-0.241-0.141—   
chr17_19649022_G_Cchr17:19649022-0.403-0.279-0.306—   
chr17_19649028_T_Cchr17:19649028-0.403-0.173-0.129—   
chr17_19649026_C_Tchr17:19649026-0.399-0.401-0.176—   
chr17_19648986_C_Achr17:19648986-0.396-0.261-0.306—   
chr17_19648791_G_Cchr17:19648791-0.393-0.269-0.200<0.001%
chr17_19648795_G_Achr17:19648795-0.393-0.0660.035<0.001%
chr17_19648798_G_Achr17:196487980.3930.650-0.047—   
chr17_19648989_G_Cchr17:196489890.3930.3250.141—   
chr17_19649026_C_Gchr17:19649026-0.393-0.404-0.018—   
chr17_19648904_A_Tchr17:19648904-0.389-0.419-0.200—   
chr17_19648979_T_Achr17:19648979-0.389-0.218-0.071—   
chr17_19648995_C_Gchr17:196489950.3890.3270.082—   
chr17_19648792_G_Achr17:19648792-0.386-0.157-0.353—   
chr17_19648788_A_Cchr17:19648788-0.383-0.231-0.094—   
chr17_19649011_T_Achr17:196490110.3830.3910.082—   
chr17_19648920_C_Tchr17:19648920-0.379-0.239-0.024—   
chr17_19648924_C_Tchr17:196489240.3790.1550.129—   
chr17_19648925_C_Achr17:196489250.3790.1600.118—   
chr17_19649030_T_Cchr17:19649030-0.379-0.246-0.129—   
chr17_19649027_C_Gchr17:19649027-0.376-0.3760.012—   
chr17_19649030_T_Achr17:19649030-0.376-0.188-0.141—   
chr17_19648926_A_Gchr17:196489260.3730.0910.106—   
chr17_19648936_G_Cchr17:196489360.3730.211-0.176—   
chr17_19648976_A_Tchr17:19648976-0.373-0.266-0.224—   
chr17_19648986_C_Tchr17:19648986-0.373-0.117-0.282—   
chr17_19648907_T_Gchr17:19648907-0.366-0.355-0.106—   
chr17_19648945_C_Gchr17:196489450.3660.2390.118—   
chr17_19649021_C_Achr17:196490210.366-0.0510.100—   
chr17_19649026_C_Achr17:19649026-0.366-0.338-0.188—   
chr17_19649065_A_Gchr17:196490650.3630.3500.188—   
chr17_19648777_C_Tchr17:19648777-0.359-0.0580.000—   
chr17_19648896_A_Tchr17:196488960.3590.2230.176—   
chr17_19648960_C_Achr17:19648960-0.359-0.195-0.129—   
chr17_19649049_G_Cchr17:19649049-0.359-0.058-0.294—   
chr17_19649054_A_Gchr17:19649054-0.359-0.107-0.300—   
chr17_19648899_C_Gchr17:19648899-0.356-0.109-0.353—   
chr17_19649031_G_Tchr17:19649031-0.356-0.226-0.165—   
chr17_19648817_C_Gchr17:19648817-0.353-0.2340.094<0.001%
chr17_19648843_T_Achr17:19648843-0.353-0.1170.082—   
chr17_19648845_T_Gchr17:19648845-0.353-0.137-0.047—   
chr17_19648847_G_Cchr17:196488470.3530.1520.059—   
chr17_19648868_C_Achr17:19648868-0.353-0.287-0.129<0.001%
chr17_19648938_C_Achr17:196489380.3530.1730.129—   
chr17_19649068_A_Gchr17:196490680.3530.3580.365—   
chr17_19648956_T_Achr17:196489560.3490.2660.306—   
chr17_19648828_C_Tchr17:19648828-0.346-0.157-0.224—   
chr17_19648901_T_Gchr17:19648901-0.343-0.175-0.224—   
chr17_19648798_G_Cchr17:196487980.3390.109-0.094—   
chr17_19648834_A_Cchr17:196488340.3390.1070.012—   
chr17_19648848_G_Tchr17:196488480.3390.147-0.1410.0013%
chr17_19648860_G_Achr17:196488600.3390.0910.024—   
chr17_19648884_G_Cchr17:196488840.3390.1350.306—   
chr17_19648907_T_Cchr17:19648907-0.339-0.373-0.118<0.001%
chr17_19648926_A_Cchr17:19648926-0.060-0.107-0.600—   
chr17_19649022_G_Achr17:196490220.3390.3350.135—   
chr17_19648883_G_Achr17:19648883-0.336-0.122-0.200—   
chr17_19649030_T_Gchr17:19649030-0.336-0.188-0.047—   
chr17_19648784_A_Cchr17:196487840.3330.0380.235—   
chr17_19648804_G_Cchr17:19648804-0.333-0.261-0.118—   
chr17_19648860_G_Tchr17:196488600.3330.2080.235—   
chr17_19648901_T_Cchr17:19648901-0.333-0.216-0.212—   
chr17_19649031_G_Cchr17:19649031-0.333-0.226-0.100—   
chr17_19648774_T_Gchr17:19648774-0.329-0.051-0.106—   
chr17_19648923_C_Tchr17:196489230.3290.1730.0940.0013%
chr17_19649079_G_Tchr17:196490790.3290.0280.235—   
chr17_19648803_C_Gchr17:19648803-0.326-0.4010.129—   
chr17_19648847_G_Tchr17:196488470.3260.1680.000—   
chr17_19648927_C_Achr17:196489270.3260.1930.188—   
chr17_19648908_G_Achr17:19648908-0.323-0.312-0.106—   
chr17_19648997_G_Cchr17:19648997-0.323-0.312-0.229—   
chr17_19648779_G_Cchr17:196487790.3190.1800.200—   
chr17_19648780_T_Gchr17:19648780-0.319-0.0180.000<0.001%
chr17_19648832_T_Gchr17:19648832-0.319-0.1980.047—   
chr17_19648908_G_Tchr17:19648908-0.319-0.332-0.235—   
chr17_19648962_G_Tchr17:196489620.3190.2230.165—   
chr17_19648897_G_Tchr17:19648897-0.316-0.185-0.294—   
chr17_19648943_G_Tchr17:196489430.3160.0330.141—   
chr17_19648809_T_Gchr17:19648809-0.313-0.2280.141—   
chr17_19648895_G_Achr17:19648895-0.313-0.203-0.176—   
chr17_19648905_C_Achr17:19648905-0.313-0.419-0.306—   
chr17_19648773_C_Gchr17:19648773-0.309-0.112-0.012—   
chr17_19648881_G_Cchr17:19648881-0.309-0.221-0.094<0.001%
chr17_19648892_G_Achr17:19648892-0.309-0.170-0.329—   
chr17_19649015_G_Cchr17:196490150.3090.2590.200—   
chr17_19648797_G_Achr17:196487970.3060.4570.071—   
chr17_19648833_G_Cchr17:196488330.3060.1520.188—   
chr17_19648866_C_Gchr17:196488660.306-0.0890.118—   
chr17_19648943_G_Cchr17:196489430.3060.1650.176—   
chr17_19648963_G_Cchr17:196489630.3060.2230.082—   

Showing 200 of 200 in this window. Scores are the p99-scaled [−1, 1] value; click a column to sort.