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UGT1A4

receptor: PXRTier 1

Drug substrates

lamotrigine; olanzapine; imipramine

refs: 25275310, 40301309

CAMIP causal chains

PXR

Blunted receptor-mediated induction of UGT1A4, leading to attenuated clearance and increased systemic exposure of its clinical substrates such as lamotrigine.

Affected substrate drugs (PharmGKB): lamotrigine; tamoxifen; ABT-751; anastrozole; testosterone

Scored variants near UGT1A4

chr2:233,618,735..233,873,300, gene body plus 100 kb. Showing the strongest 200 by effect size.

VariantPosition PXR FXR AhR AF
chr2_233718647_A_Tchr2:23371864751,39214,20824,832—   
chr2_233718667_T_Gchr2:233718667-50,048-17,024-36,352—   
chr2_233691696_G_Tchr2:23369169648,3849,02446,400—   
chr2_233718674_T_Gchr2:233718674-47,744-17,168-35,200—   
chr2_233718675_A_Tchr2:233718675-45,760-14,432-36,736—   
chr2_233718658_G_Cchr2:233718658-45,056-15,328-34,560—   
chr2_233718677_T_Gchr2:233718677-44,992-16,128-41,216—   
chr2_233718674_T_Cchr2:233718674-43,456-14,128-28,800—   
chr2_233718681_T_Achr2:233718681-42,176-14,192-35,328—   
chr2_233718675_A_Cchr2:233718675-42,112-12,656-31,232—   
chr2_233718621_T_Gchr2:233718621-41,280-12,736-27,008—   
chr2_233718557_G_Cchr2:23371855740,57612,28817,792—   
chr2_233718666_T_Achr2:233718666-40,128-14,960-27,520—   
chr2_233718681_T_Gchr2:233718681-40,064-12,848-29,568—   
chr2_233718665_A_Cchr2:233718665-39,872-12,400-25,856—   
chr2_233718659_T_Cchr2:233718659-39,360-12,512-31,232—   
chr2_233718682_A_Cchr2:233718682-39,104-13,408-31,232—   
chr2_233718670_T_Gchr2:233718670-37,120-12,096-23,552—   
chr2_233718659_T_Gchr2:233718659-37,056-12,048-29,056—   
chr2_233718647_A_Gchr2:23371864736,0329,69617,664—   
chr2_233718674_T_Achr2:233718674-35,648-11,792-24,320—   
chr2_233718662_T_Achr2:23371866235,58413,50416,768—   
chr2_233718644_C_Gchr2:23371864435,0088,57621,248—   
chr2_233718677_T_Achr2:233718677-34,880-12,576-30,080—   
chr2_233718649_C_Achr2:233718649-34,752-9,632-26,496—   
chr2_233718667_T_Achr2:233718667-34,240-11,984-20,864—   
chr2_233718683_A_Tchr2:233718683-34,240-11,488-29,056—   
chr2_233691675_A_Cchr2:23369167534,1449,37627,520—   
chr2_233718681_T_Cchr2:233718681-34,048-12,096-28,544—   
chr2_233718675_A_Gchr2:233718675-33,920-11,408-24,576—   
chr2_233718663_A_Tchr2:23371866333,2806,75217,152—   
chr2_233718710_T_Gchr2:23371871031,93610,04820,480—   
chr2_233718672_G_Cchr2:233718672-31,168-10,976-20,736—   
chr2_233718649_C_Gchr2:233718649-30,976-9,584-22,144—   
chr2_233718601_G_Achr2:23371860130,8489,72812,928—   
chr2_233718682_A_Gchr2:233718682-30,592-10,592-23,552—   
chr2_233718704_T_Cchr2:23371870430,46410,14416,384—   
chr2_233718703_C_Gchr2:23371870329,5687,90416,512—   
chr2_233718555_G_Cchr2:23371855529,0569,50413,824—   
chr2_233718625_T_Achr2:23371862529,0568,89614,848—   
chr2_233718659_T_Achr2:233718659-28,800-9,904-22,528—   
chr2_233718658_G_Achr2:233718658-28,480-9,488-18,176—   
chr2_233718677_T_Cchr2:233718677-28,096-9,488-21,632—   
chr2_233718683_A_Cchr2:233718683-27,904-9,808-22,912—   
chr2_233718682_A_Tchr2:233718682-27,264-9,088-20,736—   
chr2_233718575_C_Tchr2:23371857527,1366,7209,600—   
chr2_233718665_A_Gchr2:233718665-27,136-8,672-16,384—   
chr2_233718684_C_Tchr2:233718684-26,816-10,096-25,984—   
chr2_233718710_T_Cchr2:23371871026,5608,28816,896—   
chr2_233718676_A_Gchr2:233718676-26,304-9,760-25,600—   
chr2_233718696_A_Tchr2:233718696-26,304-8,400-18,176—   
chr2_233718666_T_Cchr2:233718666-26,240-9,632-16,512—   
chr2_233718658_G_Tchr2:233718658-26,112-8,864-17,152—   
chr2_233718663_A_Cchr2:23371866325,9844,73615,744—   
chr2_233718668_A_Tchr2:233718668-25,152-7,712-17,536—   
chr2_233718676_A_Cchr2:233718676-24,512-8,080-21,504—   
chr2_233718602_C_Gchr2:23371860224,1927,58410,112—   
chr2_233718666_T_Gchr2:233718666-24,128-8,832-14,848—   
chr2_233691757_C_Achr2:23369175723,9044,00020,096—   
chr2_233718691_A_Gchr2:233718691-23,744-7,792-15,232—   
chr2_233718684_C_Achr2:233718684-23,552-9,040-23,040—   
chr2_233718709_A_Gchr2:23371870923,1688,41614,976—   
chr2_233718671_G_Achr2:23371867122,9125,7928,448—   
chr2_233718544_A_Tchr2:23371854422,6566,62410,112—   
chr2_233718621_T_Achr2:233718621-22,528-6,720-14,720—   
chr2_233718678_A_Tchr2:233718678-22,208-8,224-19,200—   
chr2_233718694_G_Cchr2:233718694-22,208-7,136-13,696—   
chr2_233718707_C_Tchr2:233718707-22,208-7,536-15,360—   
chr2_233718683_A_Gchr2:233718683-22,144-7,344-16,896—   
chr2_233718575_C_Gchr2:23371857522,0163,9047,808—   
chr2_233718710_T_Achr2:23371871021,9525,44015,232—   
chr2_233718594_C_Achr2:233718594-21,888-7,136-13,312—   
chr2_233718591_G_Tchr2:233718591-21,824-6,880-13,056—   
chr2_233718619_G_Achr2:233718619-21,696-6,576-12,800—   
chr2_233718605_T_Achr2:23371860521,6324,5768,064—   
chr2_233718705_T_Gchr2:23371870521,6325,47211,136—   
chr2_233718638_T_Gchr2:233718638-21,376-5,952-13,696—   
chr2_233718673_G_Tchr2:23371867321,3763,2646,016—   
chr2_233718601_G_Cchr2:23371860120,9928,35212,544—   
chr2_233718650_G_Cchr2:23371865020,9286,9769,600—   
chr2_233718667_T_Cchr2:233718667-20,928-9,248-13,184—   
chr2_233718697_C_Achr2:233718697-20,928-6,912-13,056—   
chr2_233718696_A_Cchr2:233718696-20,864-6,336-13,696—   
chr2_233718684_C_Gchr2:233718684-20,544-7,360-18,304—   
chr2_233718693_G_Tchr2:23371869320,5447,52010,752—   
chr2_233718711_T_Cchr2:23371871120,4167,58414,208—   
chr2_233718593_T_Gchr2:233718593-20,160-7,136-12,160—   
chr2_233718591_G_Cchr2:233718591-19,968-6,016-11,648—   
chr2_233718649_C_Tchr2:233718649-19,648-6,240-14,848—   
chr2_233718597_A_Gchr2:23371859719,5847,00811,520—   
chr2_233718670_T_Achr2:233718670-19,520-5,696-11,648—   
chr2_233718665_A_Tchr2:233718665-19,328-4,000-12,672—   
chr2_233718643_C_Achr2:23371864319,2644,4168,320—   
chr2_233718656_C_Achr2:233718656-18,944-5,536-13,312—   
chr2_233718672_G_Achr2:233718672-18,688-6,528-12,032—   
chr2_233718622_T_Gchr2:233718622-18,624-5,920-12,288—   
chr2_233718695_C_Gchr2:23371869518,6247,13612,544—   
chr2_233718577_C_Achr2:233718577-18,560-5,472-9,984—   
chr2_233718646_T_Achr2:23371864618,4325,76011,392—   
chr2_233718713_C_Tchr2:233718713-18,432-6,768-13,440—   
chr2_233718595_A_Tchr2:233718595-18,240-6,208-12,928—   
chr2_233718591_G_Achr2:233718591-18,176-5,728-11,264—   
chr2_233718661_A_Cchr2:233718661-17,984-5,792-12,800—   
chr2_233718706_C_Gchr2:23371870617,9844,5763,968—   
chr2_233718569_A_Cchr2:23371856917,7925,0568,576—   
chr2_233718672_G_Tchr2:233718672-17,728-5,632-11,392—   
chr2_233718645_A_Gchr2:23371864517,6644,76810,624—   
chr2_233718567_G_Cchr2:233718567-17,280-5,248-8,192—   
chr2_233718593_T_Achr2:233718593-17,280-6,144-11,136—   
chr2_233718668_A_Cchr2:233718668-17,216-6,320-12,032—   
chr2_233718545_T_Achr2:23371854517,1525,9849,728—   
chr2_233718595_A_Gchr2:233718595-16,960-5,536-9,600—   
chr2_233718696_A_Gchr2:233718696-16,960-5,824-11,520—   
chr2_233718680_G_Cchr2:233718680-16,704-5,504-12,928—   
chr2_233718686_G_Achr2:23371868616,5764,7689,088—   
chr2_233718712_A_Gchr2:23371871216,3205,20011,008—   
chr2_233718711_T_Gchr2:23371871116,2564,51210,752—   
chr2_233718565_T_Achr2:233718565-16,192-5,632-9,344—   
chr2_233718579_G_Tchr2:233718579-16,192-5,216-9,472—   
chr2_233718661_A_Tchr2:233718661-16,192-4,672-12,544—   
chr2_233718655_G_Tchr2:23371865516,0005,5687,552—   
chr2_233718577_C_Tchr2:233718577-15,808-5,248-11,136—   
chr2_233691687_C_Gchr2:23369168715,7765,08814,464—   
chr2_233718651_A_Tchr2:233718651-15,616-5,312-9,472—   
chr2_233718669_A_Gchr2:233718669-15,616-7,264-8,960—   
chr2_233718596_G_Cchr2:23371859615,4245,8569,984—   
chr2_233718574_C_Gchr2:23371857415,3604,5126,528—   
chr2_233718620_A_Tchr2:23371862015,3605,1524,992—   
chr2_233718637_T_Achr2:233718637-15,360-4,960-9,856—   
chr2_233718654_G_Tchr2:233718654-15,360-4,960-10,624—   
chr2_233718605_T_Cchr2:233718605-15,296-4,960-8,320—   
chr2_233718646_T_Gchr2:23371864615,1684,7368,320—   
chr2_233718685_T_Gchr2:233718685-15,104-5,440-8,448—   
chr2_233718695_C_Achr2:23371869515,0405,2488,960—   
chr2_233718567_G_Achr2:233718567-14,592-4,576-8,448—   
chr2_233718629_T_Achr2:233718629-14,528-4,416-9,344—   
chr2_233718643_C_Tchr2:23371864314,5284,0965,632—   
chr2_233718663_A_Gchr2:233718663-14,528-4,576-8,704—   
chr2_233718547_A_Tchr2:23371854714,3364,8968,064—   
chr2_233718553_A_Cchr2:23371855314,2724,1287,040—   
chr2_233718641_G_Cchr2:23371864114,1444,0006,272—   
chr2_233718669_A_Cchr2:233718669-14,080-6,304-6,656—   
chr2_233718673_G_Cchr2:23371867314,0162,9766,016—   
chr2_233718678_A_Cchr2:23371867813,9523,76010,624—   
chr2_233718623_G_Cchr2:233718623-13,824-3,360-9,472—   
chr2_233718592_G_Tchr2:233718592-13,632-4,576-8,704—   
chr2_233718697_C_Tchr2:233718697-13,568-4,960-8,064—   
chr2_233718709_A_Cchr2:23371870913,3765,08810,752—   
chr2_233718611_A_Gchr2:23371861112,9924,73610,496—   
chr2_233718712_A_Cchr2:23371871212,9923,50410,112—   
chr2_233718671_G_Cchr2:23371867112,8003,3926,656—   
chr2_233718713_C_Gchr2:233718713-12,736-5,040-10,112—   
chr2_233718594_C_Gchr2:233718594-12,672-4,512-7,936—   
chr2_233718650_G_Tchr2:233718650-12,608-3,392-9,984—   
chr2_233718679_A_Cchr2:233718679-12,544-3,712-7,808—   
chr2_233718685_T_Achr2:233718685-12,544-4,096-9,216—   
chr2_233718563_A_Tchr2:233718563-12,288-3,808-7,552—   
chr2_233718644_C_Tchr2:233718644-12,288-4,448-7,168—   
chr2_233718630_C_Gchr2:23371863012,2242,6887,296—   
chr2_233718708_A_Tchr2:23371870812,2243,5689,600—   
chr2_233718691_A_Tchr2:233718691-12,160-4,448-7,936—   
chr2_233718711_T_Achr2:23371871112,1602,9767,552—   
chr2_233718573_T_Gchr2:23371857312,0323,6166,272—   
chr2_233718606_T_Cchr2:23371860612,0323,3924,736—   
chr2_233718699_T_Achr2:233718699-12,032-4,352-8,192—   
chr2_233718592_G_Achr2:233718592-11,968-3,680-7,936—   
chr2_233718577_C_Gchr2:233718577-11,904-3,232-4,608—   
chr2_233718553_A_Tchr2:23371855311,8403,2965,760—   
chr2_233718594_C_Tchr2:233718594-11,840-4,416-7,552—   
chr2_233718600_A_Cchr2:233718600-11,776-4,352-5,376—   
chr2_233718639_G_Tchr2:23371863911,7762,3044,096—   
chr2_233718601_G_Tchr2:23371860111,6484,2245,760—   
chr2_233718629_T_Cchr2:233718629-11,584-3,520-6,784—   
chr2_233718631_C_Gchr2:233718631-11,584-3,552-7,296—   
chr2_233718618_T_Achr2:233718618-11,456-3,520-6,912—   
chr2_233718687_G_Achr2:233718687-11,200-3,488-5,376—   
chr2_233718608_A_Gchr2:23371860811,0082,6246,656—   
chr2_233718653_A_Cchr2:23371865311,0082,6886,144—   
chr2_233718662_T_Cchr2:23371866211,0085,0566,400—   
chr2_233718679_A_Gchr2:233718679-11,008-2,928-6,016—   
chr2_233718626_C_Tchr2:23371862610,9443,8725,248—   
chr2_233718566_T_Achr2:233718566-10,880-3,680-6,912—   
chr2_233718588_C_Gchr2:233718588-10,688-3,936-7,040—   
chr2_233718616_C_Tchr2:233718616-10,688-3,616-8,704—   
chr2_233718590_G_Achr2:23371859010,6242,9125,248—   
chr2_233718595_A_Cchr2:233718595-10,624-3,520-4,096—   
chr2_233718597_A_Cchr2:23371859710,6243,4246,016—   
chr2_233718680_G_Achr2:233718680-10,624-4,208-9,472—   
chr2_233718599_G_Achr2:23371859910,4962,4003,584—   
chr2_233718679_A_Tchr2:233718679-10,496-2,464-6,272—   
chr2_233718631_C_Tchr2:233718631-10,368-3,072-7,424—   
chr2_233718618_T_Cchr2:233718618-10,304-3,840-4,480—   
chr2_233718702_T_Gchr2:23371870210,3043,6166,016—   
chr2_233718633_A_Cchr2:23371863310,2404,3205,632—   
chr2_233718680_G_Tchr2:23371868010,2401,7926,144—   
chr2_233691648_T_Achr2:233691648-9,408-3,680-11,456—   
chr2_233691723_C_Gchr2:233691723-8,448-3,040-10,816—   
chr2_233691664_G_Tchr2:233691664-8,256-2,656-10,304—   
chr2_233691696_G_Cchr2:2336916966,9121,76010,624—   
chr2_233691682_T_Gchr2:2336916824,0321,72810,688—   

Showing 200 of 200 in this window. Scores are the raw center bin Δ, ALT minus REF; click a column to sort.